Detalhes da Produção

TipoPatente
GrupoProdução Técnica
DescriçãoROMEIRO, L. A. S. ; FRAGA, Carlos Alberto Manssour ; BARREIRO, Eliezer Jesus de Lacerda ; SILVA, Cláudia Lúcia Martins da ; MIRANDA, Ana Luisa Palhares de ; BRITO, Fernanda Carla Ferreira de ; ALMEIDA, Helena Carla Castro Cardoso de ; NOËL, François Germain ; TIBIRIÇÁ, Eduardo Vera, Use of Adrenergic N-Phenylpiperazine Antagonists, Pharmaceutical Compositions Containning Them, and Methods of Preparing Them. 2007, Estados Unidos.
AutorLuiz Antonio Soares Romeiro
Ano2007

Informações Complementares

Ano de Desenvolvimento2007
Codigo do Registro ou PatenteUS2007219213
Data Pedido de Deposito20/09/2007
FinalidadeBenign prostatic hyperplasia
Informações AdicionaisAbstract of Patent Application US2007219213 The present invention describes phenylpiperazinyl alpha adrenergic antagonists that corresponds to the formula (I) which selectively act on the alpha 1A/alpha 1D subtypes, where its selectivity index in comparison to alpha 1B subtype is, at minimum, 1700 for the alpha 1A subtype and 10000 for the alpha 1 D subtype, being therefore useful for the treatment of the lower urinary tract symptoms, including the benign prostatic hyperplasia treatment in mammals, preferentially humans. It is also described pharmaceutical compositions containing said compounds and methods for its preparation.
Instituição FinanciadoraUBEC
Meio de DivulgaçãoIMPRESSO
PaísEstados Unidos
Potencial de InovaçãoNAO
RelevânciaNAO
Tipo de PatentePATENTE_NO_EXTERIOR_PE
TítuloUse of Adrenergic N-Phenylpiperazine Antagonists, Pharmaceutical Compositions Containning Them, and Methods of Preparing Them
Título da PatenteUse of Adrenergic N-Phenylpiperazine Antagonists, Pharmaceutical Compositions Containning Them, and Methods of Preparing Them