Detalhes da Produção

TipoDesenho Industrial
GrupoProdução Técnica
DescriçãoROMEIRO, L. A. S.. Use Of Adrenergic N-Phenylpiperazine Antagonists, Pharmaceutical Compositions Containing Them, And Methods Of Preparing Them. 2005, Brasil. Patente: Desenho Industrial. Número do registro: WO2005/112538A2, data de registro: 01122005, título: "Use Of Adrenergic N-Phenylpiperazine Antagonists, Pharmaceutical Compositions Containing Them, And Methods Of Preparing Them" . Instituição(ões) financiadora(s): UFRJ / UBEC.
AutorLuiz Antonio Soares Romeiro
Ano2005

Informações Complementares

Ano de Desenvolvimento2005
descricao-informacoes-adicionaisPCT WO 2005/112538 - Abstract The present invention describes phenylpiperazinyl alpha adrenergic antagonists that corresponds to the formula which selectively act on the alpha 1A/alpha 1D subtypes, where its selectivity index in comparison to alpha 1B subtype is, at minimum, 1700 for the alpha 1A subtype and 10000 for the alpha 1D subtype, being therefore useful for the treatment of the lower urinary tract symptoms, including the benign prostatic hyperplasia treatment in mammals, preferentially humans. It is also described pharmaceutical compositions containing said compounds and methods for its preparation.
FinalidadeTratamento de sintomas do trato urinário inferior
flag-potencial-inovacaoNAO
instituicao-financiadoraUFRJ / UBEC
PaísBrasil
RelevânciaNAO
TítuloUse Of Adrenergic N-Phenylpiperazine Antagonists, Pharmaceutical Compositions Containing Them, And Methods Of Preparing Them
DDMMAAAA
DESENHO_INDUSTRIAL_DI
WO2005/112538A2
Use Of Adrenergic N-Phenylpiperazine Antagonists, Pharmaceutical Compositions Containing Them, And Methods Of Preparing Them
01122005